Antidepressant Tianeptine Sodium Salt Powder CAS 30123-17-2 White Color

Place of Origin CHINA
Brand Name XRD
Certification GMP
Model Number 30123-17-2
Minimum Order Quantity negotiable
Price Inquiry for Negotiable
Packaging Details 1-2 Kg / Aluminum Foil Bag, 25kg/ Drum, as Require
Delivery Time 1-2days after payment received
Payment Terms T/T, Western Union,Bitcoin
Supply Ability 5000kg/year

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Product Details
Cas No. 30123-17-2 Other Names S-1574
Product NamRopivacainee Tianeptine Sodium Salt Appearance White Powder
Assay 99% Tianeptine Sodium Salt Grade Pharmaceutical Grade
Storage Cool Dried Storage Application Pharmaceutical Raw Intermediates
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Product Description

Antidepressant Tianeptine Sodium Salt Powder CAS 30123-17-2 White Color

Description:

 

Tianeptine sodium salt is a salt of Tianeptine. Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake . Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation.

 

 

COA: 

 

Description

White to yellowish powder,very hygroscopic.

Solubility

Freetly soluble In water and methanol and dichloromethane

Identification

(1)By IR, To match with working standard

(2)It gives reaction of sodium

Related compounds

Any impurity ≤0.1%
Total impurities ≤0.4%

Residual Solvents

Acetidin≤ 0.5%
Dichloromethane≤ 0.06%
Methanol 0.3%
Acetone 0.5%
Acetonitrile≤0.041%
Ethanol≤0.5%
N, N-dimethylformamide ≤0.088%
Water ≤ 5.0%

Assay

99.0%-101.0%(On anhydrous basis)
 

 

Function: 

 

Tianeptine is antidepressant. The animal has: the hippocampus pyramidal cells increased spontaneous activity, and accelerating its function was inhibited after recovery; increase in cortical and hippocampal neurons at sites of 5- serotonin reuptake. Tianeptine without following adverse effects: sleep and alertness; cardiovascular system; cholinergic system ( without anticholinergic symptoms ); drug craving.

 

 

Applicaiton: 

 

Tianeptine has antidepressant and anxiolytic (anti-anxiety) properties with a relative lack of sedative, anticholinergic and cardiovascular adverse effects, thus suggesting it is particularly suitable for use in the elderly and in those following alcohol withdrawal; such persons can be more sensitive to the adverse effects of psychotropic drugs. Recent results indicate possible anticonvulsant (anti-seizure) and analgesic (painkilling) activity of tianeptine via immediate or downstream modulation of adenosine A1 receptors (as the effects could be experimentally blocked by antagonists of this receptor).

 

 

 

Antidepressant Tianeptine Sodium Salt Powder CAS 30123-17-2 White Color 0

 

 

 

Packing:

 

1

 

 

Antidepressant Tianeptine Sodium Salt Powder CAS 30123-17-2 White Color